H
N
HN
O
O
NCL1
O
NH 2
PCPA
NH 2
NCD38
HN
O
O
NH
Cl
H
N
H
N
GSK2879552
H
N
ORY-1001
NH 2
N
COOH
NH 2
H
N
O
N
N
Me
1
N
N
O
OMe
N
H
O
NH 2
2
N
OH
O
NH
NH 2
3
O
O
N Me
N
O
N
Me
Me
R
PCPA-Tamoxifen Conjugates (R = H, Me)
N
Me
pargyline
O
OH H
N
T5342129
Fig. 2 Examples of LSD1 inhibitors
204
T. Suzuki