140
M. M. Kabanda and K. P. Otukile
3. Tanabe Y, Suzukamo G, Komuro Y, Imanishi N, Morooka S, Enomoto M, Kojima A,
Sanemitsu Y, Mizutani M (1991) Structure-activity relationship of optically active 2-(3pyridyl)thiazolidin-4-ones as a PAF antagonists. Tetrahedron Lett 32:379–382
4. Rawal RK, Prabhakar YS, Katti SB, De Clercq E (2005) 2-(Aryl)-3-furan-2-ylmethylthiazolidin-4-ones as selective HIV-RT Inhibitors. Bioorg Med Chem 13:6771–6776
5. Srivastava T, Gaikwad AK, Haq W (2005) Synthesis and biological evaluation of 4thiazolidinone derivatives as potential antimycobacterial agents. Arkivoc ii: 120–130
6. Rajopadhye M, Popp FD (1987) Synthesis and antileukemic activity of spiro[indoline-3,2 -
thiazolidine]-2,4 -diones. J Heterocyclic Chem 24:1637–1642
7. Metwally NH, Radwan IT, El-Serwy WS, Mohamed MA (2019) Design, synthesis, DNA
assessment and molecular docking study of novel 2-(pyridin-2-ylimino)thiazolidin-4-one
derivatives as potent antifungal agents. Bioorg Chem 84:456–467
8. Pan B, Huang R-Z, Han S-Q (2010) Design, synthesis, and antibiofilm activity of 2-arylimino3-aryl-thiazolidine-4-ones. Bioorg Med Chem Lett 20:2461–2464
9. El-Gazzar A-RBA, Gaffar MA-E-D, Ali SA (2008) Design, synthesis, and preliminary evaluation as antimicrobial activity of novel spiro-1, 3-thiazolidine C-acyclic nucleoside analogs. J
Sulfur Chem 29:549–558
10. Nagalakshmi G, Maity TK, Maiti BC (2013) Synthesis, characterization and antiviral evaluation
of some novel 2-[(substitutedphenyl/heteroaryl)imino]-3-phenyl-1,3- thiazolidin-4-ones. Der
Pharmacia Lett 5:177–188
11. Bolli MH, Abele S, Binkert C, Bravo R, Buchmann S, Bur D, Gatfield J, Hess P, Kohl C,
Mangold C, Mathys B, Menyhart K, Müller C, Nayler O, Scherz M, Schmidt G, Sippel V,
Steiner B, Strasser D, Treiber A, Weller T (2010) 2-imino-thiazolidin-4-one derivatives as
potent, orally active S1P1 receptor agonists. J Med Chem 53:4198–4211
12. Akerblom E (1967) 2-aminothiazolidin-4-one and 2-iminothiazolidin-4-one. Part I. The
reaction of chloroacetic acid with N-monoalkylthiurea. Acta Chim Scand 21:843–848
13. Kasmi-Mir S, Djafri A, Paquin L, Hamelin J, Rahmouni M (2006) One-pot synthesis of 5arylidene-2-imino-4-thiazolidinones under microwave irradiation. Molecules 11:597–602
14. Sathishkumar M, Nagarajan S, Shanmugavelan P, Dinesh M, Ponnuswamy A (2013) A
facile, rapid, one-pot regio/stereoselective synthesis of 2-iminothiazolidin-4-ones under
solvent/scavenger-free conditions. Beilstain J Org Chem 9:689–697
15. Meng G, Zheng M, Dong M, Qu Q (1998) An eco-friendly preparation of 2-iminothiazolidin4-ones derivatives. Org Prep Proced Int 44:184–186
16. Kasmi S, Hamelin J, Benhaoua H (1998) Microwave-assisted solvent-free synthesis of
iminothiazolines. Tetrahedron Lett 39:8093–8096
17. Murru S, Singh CB, Kavala V (2008) A convenient one-pot synthesis of thiazol-2-imines:
application in the construction of pifithrin analogues. Tetrahedron 64:1931–1942
18. Meng G, Li ZY, Zheng ML (2008) An efficient one-step method for the large-scale synthesis
of 2,4-thiazolidinedione. Org Prep Proced Int 40:572–574
19. Meng G, Gao Y, Zheng ML (2011) Improved preparation of 2,4-thiazolidinedione. Org Prep
Proced Int 43:312–313
20. Lynch BJ, Truhlar DG (2001) How well can hybrid density functional methods predict transition
sate geometries and barrier heights? J Phys Chem A 105:2936–2941
21. Zhao Y, Schultz NE, Truhlar DG (2006) Design of density functionals by combining the method
of constraint satisfaction with parametrization for thermochemistry, thermochemical kinetics,
and noncovalent interactions. J Chem Theory Comput 2:364–382
22. Zhao Y, Truhlar DG (2008) Exploring the limit of accuracy of the global hybrid meta density
functional for main-group thermochemistry, kinetics, and noncovalent interactions. J Chem
Theory Comput 4:1849–1868
23. Marenich AV, Cramer CJ, Truhlar DG (2009) Universal solvation model based on solute electron density and a continuum model of the solvent defined by the bulk dielectric constant and
atomic surface tensions. J Phys Chem B 113:6378–6396
24. Peverati R, Truhlar DG (2014) The quest for a universal density functional: the accuracy of
density functionals across a broad spectrum of databases in chemistry and physics. Phil Trans
R Soc A 372: 20120476/1-51
M. M. Kabanda and K. P. Otukile
3. Tanabe Y, Suzukamo G, Komuro Y, Imanishi N, Morooka S, Enomoto M, Kojima A,
Sanemitsu Y, Mizutani M (1991) Structure-activity relationship of optically active 2-(3pyridyl)thiazolidin-4-ones as a PAF antagonists. Tetrahedron Lett 32:379–382
4. Rawal RK, Prabhakar YS, Katti SB, De Clercq E (2005) 2-(Aryl)-3-furan-2-ylmethylthiazolidin-4-ones as selective HIV-RT Inhibitors. Bioorg Med Chem 13:6771–6776
5. Srivastava T, Gaikwad AK, Haq W (2005) Synthesis and biological evaluation of 4thiazolidinone derivatives as potential antimycobacterial agents. Arkivoc ii: 120–130
6. Rajopadhye M, Popp FD (1987) Synthesis and antileukemic activity of spiro[indoline-3,2 -
thiazolidine]-2,4 -diones. J Heterocyclic Chem 24:1637–1642
7. Metwally NH, Radwan IT, El-Serwy WS, Mohamed MA (2019) Design, synthesis, DNA
assessment and molecular docking study of novel 2-(pyridin-2-ylimino)thiazolidin-4-one
derivatives as potent antifungal agents. Bioorg Chem 84:456–467
8. Pan B, Huang R-Z, Han S-Q (2010) Design, synthesis, and antibiofilm activity of 2-arylimino3-aryl-thiazolidine-4-ones. Bioorg Med Chem Lett 20:2461–2464
9. El-Gazzar A-RBA, Gaffar MA-E-D, Ali SA (2008) Design, synthesis, and preliminary evaluation as antimicrobial activity of novel spiro-1, 3-thiazolidine C-acyclic nucleoside analogs. J
Sulfur Chem 29:549–558
10. Nagalakshmi G, Maity TK, Maiti BC (2013) Synthesis, characterization and antiviral evaluation
of some novel 2-[(substitutedphenyl/heteroaryl)imino]-3-phenyl-1,3- thiazolidin-4-ones. Der
Pharmacia Lett 5:177–188
11. Bolli MH, Abele S, Binkert C, Bravo R, Buchmann S, Bur D, Gatfield J, Hess P, Kohl C,
Mangold C, Mathys B, Menyhart K, Müller C, Nayler O, Scherz M, Schmidt G, Sippel V,
Steiner B, Strasser D, Treiber A, Weller T (2010) 2-imino-thiazolidin-4-one derivatives as
potent, orally active S1P1 receptor agonists. J Med Chem 53:4198–4211
12. Akerblom E (1967) 2-aminothiazolidin-4-one and 2-iminothiazolidin-4-one. Part I. The
reaction of chloroacetic acid with N-monoalkylthiurea. Acta Chim Scand 21:843–848
13. Kasmi-Mir S, Djafri A, Paquin L, Hamelin J, Rahmouni M (2006) One-pot synthesis of 5arylidene-2-imino-4-thiazolidinones under microwave irradiation. Molecules 11:597–602
14. Sathishkumar M, Nagarajan S, Shanmugavelan P, Dinesh M, Ponnuswamy A (2013) A
facile, rapid, one-pot regio/stereoselective synthesis of 2-iminothiazolidin-4-ones under
solvent/scavenger-free conditions. Beilstain J Org Chem 9:689–697
15. Meng G, Zheng M, Dong M, Qu Q (1998) An eco-friendly preparation of 2-iminothiazolidin4-ones derivatives. Org Prep Proced Int 44:184–186
16. Kasmi S, Hamelin J, Benhaoua H (1998) Microwave-assisted solvent-free synthesis of
iminothiazolines. Tetrahedron Lett 39:8093–8096
17. Murru S, Singh CB, Kavala V (2008) A convenient one-pot synthesis of thiazol-2-imines:
application in the construction of pifithrin analogues. Tetrahedron 64:1931–1942
18. Meng G, Li ZY, Zheng ML (2008) An efficient one-step method for the large-scale synthesis
of 2,4-thiazolidinedione. Org Prep Proced Int 40:572–574
19. Meng G, Gao Y, Zheng ML (2011) Improved preparation of 2,4-thiazolidinedione. Org Prep
Proced Int 43:312–313
20. Lynch BJ, Truhlar DG (2001) How well can hybrid density functional methods predict transition
sate geometries and barrier heights? J Phys Chem A 105:2936–2941
21. Zhao Y, Schultz NE, Truhlar DG (2006) Design of density functionals by combining the method
of constraint satisfaction with parametrization for thermochemistry, thermochemical kinetics,
and noncovalent interactions. J Chem Theory Comput 2:364–382
22. Zhao Y, Truhlar DG (2008) Exploring the limit of accuracy of the global hybrid meta density
functional for main-group thermochemistry, kinetics, and noncovalent interactions. J Chem
Theory Comput 4:1849–1868
23. Marenich AV, Cramer CJ, Truhlar DG (2009) Universal solvation model based on solute electron density and a continuum model of the solvent defined by the bulk dielectric constant and
atomic surface tensions. J Phys Chem B 113:6378–6396
24. Peverati R, Truhlar DG (2014) The quest for a universal density functional: the accuracy of
density functionals across a broad spectrum of databases in chemistry and physics. Phil Trans
R Soc A 372: 20120476/1-51