307. Hutchinson I, Stevens MFG (2007) Org Biomol Chem 5:114–120
308. Foo K, Newhouse T, Mori I, Takayama H, Baran PS (2011) Angew Chem Int Ed 50:
2716–2719
309. Setessier J, Detert H (2012) Synthesis 44:290–296
310. Leahy DK, Desai LV, Deshpande RP, Mariadass AV, Rangaswamy S, Rajagopal SK,
Madhavan L, Illendula S (2012) Org Process Res Dev 16:244–249
311. Mitchell D, Cole KP, Pollock PM, Coppert DM, Burkholder TP, Clayton JR (2012)
Org Process Res Dev 16:70–81
312. Hennessy EJ, Buchwald SL (2005) J Org Chem 70:7371–7375
313. Jensen TA, Liang X, Tanner D, Skjaerbaek N (2004) J Org Chem 69:4936–4947
314. Zhu J, Pottorf RS, Player MR (2006) Tetrahedron Lett 47:7267–7270
315. Ma Y, Margarida L, Brookes J, Makara GM, Berk SC (2004) J Comb Chem 6:426–430
316. Ruhland T, Svejgaard L, Rasmussen LK, Andersen K (2004) J Comb Chem 6:934–941
317. Pitts WJ, Vaccaro W, Huynh T, Leftheris K, Roberge JY, Barbosa J, Guo J, Brown B,
Watson A, Donaldson K, Starling GC, Kiener PA, Poss MA, Dodd JH, Barrish JC (2004)
Bioorg Med Chem Lett 14:2955–2958
318. Bettinetti L, Lo ¨ber S, Hu ¨bner H, Gmeiner P (2005) J Comb Chem 7:309–316
319. Chapman CJ, Matsuno A, Frost CG, Willis MC (2007) Chem Commun 3903–3905
320. Balraju V, Iqbal J (2006) J Org Chem 71:8954–8956
321. Scho ¨n U, Messinger J, Buchholz M, Reinecker U, Thole H, Prabhu MKS, Konda A (2005)
Tetrahedron Lett 46:7111–7115
322. Browning RG, Badarinarayana V, Mahmud H, Lovely CJ (2004) Tetrahedron 60:359–365
323. Bringmann G, Gulder T, Reichert M, Meyer F (2006) Org Lett 8:1037–1040
324. Ganton MD, Kerr MA (2007) J Org Chem 72:574–582
325. Movassaghi M, Ondrus AE (2005) Org Lett 7:4423–4426
326. Ondrus AE, Movassaghi M (2006) Tetrahedron 62:5287–5297
327. Wang Z, Wang B, Wu J (2007) J Comb Chem 9:811–817
328. Wilson RM, Thalji RK, Bergman RG, Ellman JA (2006) Org Lett 8:1745–1747
329. Ganton MD, Kerr MA (2005) Org Lett 7:4777–4779
330. Girard N, Gautier C, Malassene R, Hurvois J-P, Moinet C, Toupet L (2004) Synlett
2005–2009
331. Tietze M, Iglesias A, Merisor E, Conrad J, Klaiber I, Beifuss U (2005) Org Lett 7:1549–1552
332. Inamoto K, Katsuno M, Yoshino T, Arai Y, Hiroya K, Sakamoto T (2007) Tetrahedron 63:
2695–2711
333. Smith AB III, Ku ¨rti L, Davulcu AH, Cho YS, Ohmoto K (2007) J Org Chem 72:4611–4620
334. Ohno H, Terui T, Kitawaki T, Chida N (2006) Tetrahedron Lett 47:5747–5750
335. Huang W-S, Shakespeare WC (2007) Synthesis 2121–2124
336. Bower JF, Szeto P, Gallagher T (2007) Org Lett 9:3283–3286
337. Martin MW, Newcomb J, Nunes JJ, Bemis JE, McGowan DC, White RD, Buchanan JL,
DiMauro EF, Boucher C, Faust T, Hsieh F, Huang X, Lee JH, Schneider S, Turci SM, Zhu X
(2007) Bioorg Med Chem Lett 17:2299–2304
338. Watterson SH, Chen P, Zhao Y, Gu HH, Murali Dhar TG, Xiao Z, Ballentine SK, Shen Z,
Fleener CA, Rouleau KA, Obermeier M, Yang Z, McIntyre KW, Shuster DJ, Witmer M,
Dambach D, Chao S, Mathur A, Chen B-C, Barrish JC, Robl JA, Townsend R, Iwanowicz EJ
(2007) J Med Chem 50:3730–3742
339. Zhao M, Yin J, Huffman MA, McNamara JM (2006) Tetrahedron 62:1110–1115
340. Kanbara T, Honma A, Hasegawa K (1996) Chem Lett 1135–1136
341. Singer RA, Sadighi JP, Buchwald SL (1998) J Am Chem Soc 120:213–214
342. Sadighi JP, Singer RA, Buchwald SL (1998) J Am Chem Soc 120:4960–4976
343. Zhang X-X, Sadighi JP, Mackewitz TW, Buchwald SL (2000) J Am Chem Soc 122:
7606–7607
344. Eelkema R, Anderson HL (2008) Macromolecules 41:9930–9933
345. Jin Z, Lucht BL (2005) J Am Chem Soc 127:5586–5595
50
G.S. Lemen and J.P. Wolfe
308. Foo K, Newhouse T, Mori I, Takayama H, Baran PS (2011) Angew Chem Int Ed 50:
2716–2719
309. Setessier J, Detert H (2012) Synthesis 44:290–296
310. Leahy DK, Desai LV, Deshpande RP, Mariadass AV, Rangaswamy S, Rajagopal SK,
Madhavan L, Illendula S (2012) Org Process Res Dev 16:244–249
311. Mitchell D, Cole KP, Pollock PM, Coppert DM, Burkholder TP, Clayton JR (2012)
Org Process Res Dev 16:70–81
312. Hennessy EJ, Buchwald SL (2005) J Org Chem 70:7371–7375
313. Jensen TA, Liang X, Tanner D, Skjaerbaek N (2004) J Org Chem 69:4936–4947
314. Zhu J, Pottorf RS, Player MR (2006) Tetrahedron Lett 47:7267–7270
315. Ma Y, Margarida L, Brookes J, Makara GM, Berk SC (2004) J Comb Chem 6:426–430
316. Ruhland T, Svejgaard L, Rasmussen LK, Andersen K (2004) J Comb Chem 6:934–941
317. Pitts WJ, Vaccaro W, Huynh T, Leftheris K, Roberge JY, Barbosa J, Guo J, Brown B,
Watson A, Donaldson K, Starling GC, Kiener PA, Poss MA, Dodd JH, Barrish JC (2004)
Bioorg Med Chem Lett 14:2955–2958
318. Bettinetti L, Lo ¨ber S, Hu ¨bner H, Gmeiner P (2005) J Comb Chem 7:309–316
319. Chapman CJ, Matsuno A, Frost CG, Willis MC (2007) Chem Commun 3903–3905
320. Balraju V, Iqbal J (2006) J Org Chem 71:8954–8956
321. Scho ¨n U, Messinger J, Buchholz M, Reinecker U, Thole H, Prabhu MKS, Konda A (2005)
Tetrahedron Lett 46:7111–7115
322. Browning RG, Badarinarayana V, Mahmud H, Lovely CJ (2004) Tetrahedron 60:359–365
323. Bringmann G, Gulder T, Reichert M, Meyer F (2006) Org Lett 8:1037–1040
324. Ganton MD, Kerr MA (2007) J Org Chem 72:574–582
325. Movassaghi M, Ondrus AE (2005) Org Lett 7:4423–4426
326. Ondrus AE, Movassaghi M (2006) Tetrahedron 62:5287–5297
327. Wang Z, Wang B, Wu J (2007) J Comb Chem 9:811–817
328. Wilson RM, Thalji RK, Bergman RG, Ellman JA (2006) Org Lett 8:1745–1747
329. Ganton MD, Kerr MA (2005) Org Lett 7:4777–4779
330. Girard N, Gautier C, Malassene R, Hurvois J-P, Moinet C, Toupet L (2004) Synlett
2005–2009
331. Tietze M, Iglesias A, Merisor E, Conrad J, Klaiber I, Beifuss U (2005) Org Lett 7:1549–1552
332. Inamoto K, Katsuno M, Yoshino T, Arai Y, Hiroya K, Sakamoto T (2007) Tetrahedron 63:
2695–2711
333. Smith AB III, Ku ¨rti L, Davulcu AH, Cho YS, Ohmoto K (2007) J Org Chem 72:4611–4620
334. Ohno H, Terui T, Kitawaki T, Chida N (2006) Tetrahedron Lett 47:5747–5750
335. Huang W-S, Shakespeare WC (2007) Synthesis 2121–2124
336. Bower JF, Szeto P, Gallagher T (2007) Org Lett 9:3283–3286
337. Martin MW, Newcomb J, Nunes JJ, Bemis JE, McGowan DC, White RD, Buchanan JL,
DiMauro EF, Boucher C, Faust T, Hsieh F, Huang X, Lee JH, Schneider S, Turci SM, Zhu X
(2007) Bioorg Med Chem Lett 17:2299–2304
338. Watterson SH, Chen P, Zhao Y, Gu HH, Murali Dhar TG, Xiao Z, Ballentine SK, Shen Z,
Fleener CA, Rouleau KA, Obermeier M, Yang Z, McIntyre KW, Shuster DJ, Witmer M,
Dambach D, Chao S, Mathur A, Chen B-C, Barrish JC, Robl JA, Townsend R, Iwanowicz EJ
(2007) J Med Chem 50:3730–3742
339. Zhao M, Yin J, Huffman MA, McNamara JM (2006) Tetrahedron 62:1110–1115
340. Kanbara T, Honma A, Hasegawa K (1996) Chem Lett 1135–1136
341. Singer RA, Sadighi JP, Buchwald SL (1998) J Am Chem Soc 120:213–214
342. Sadighi JP, Singer RA, Buchwald SL (1998) J Am Chem Soc 120:4960–4976
343. Zhang X-X, Sadighi JP, Mackewitz TW, Buchwald SL (2000) J Am Chem Soc 122:
7606–7607
344. Eelkema R, Anderson HL (2008) Macromolecules 41:9930–9933
345. Jin Z, Lucht BL (2005) J Am Chem Soc 127:5586–5595
50
G.S. Lemen and J.P. Wolfe
