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195. Xie JH, Zhu SF, Zhou QL (2012) Chem Soc Rev 41:4126
196. Maire P, Deblon S, Breher F, Geier J, Böhler C, Rüegger H, Schönberg H, Grützmacher H
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197. Giacomina F, Meetsma A, Panella L, Lefort L, de Vries AHM, de Vries JG (2007) Angew
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200. Hou G, Li W, Ma M, Zhang X, Zhang X (2010) J Am Chem Soc 132:12844
201. Busscher GF, Lefort L, Cremers JGO, Mottinelli M, Wiertz RW, de Lange B, Okamura Y,
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202. Han Z, Guan YQ, Liu G, Wang R, Yin X, Zhao Q, Cong H, Dong XQ, Zhang X (2018) Org
Lett 20:6349
203. Patureau FW, Worch C, Siegler MA, Spek AL, Bolm C, Reek JNH (2012) Adv Synth Catal
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206. Cabré A, Romagnoli E, Martínez-Balart P, Verdaguer X, Riera A (2019) Org Lett 21:9709
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208. Nicholas GM, Molinski TF (2000) Tetrahedron 56:2921
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210. Harris RN, Stabler RS, Repke DB, Kress JM, Walker KA, Martin RS, Brothers JM, Ilnicka M,
Lee SW, Mirzadegan T (2010) Bioorg Med Chem Lett 20:3436
211. Ramesh P, Suman D (2018) Synthesis 50:211
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213. Xie JH, Zhu SF, Zhou QL (2011) Chem Rev 111:1713
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221. Salomó E, Rojo P, Hernández-Lladó P, Riera A, Verdaguer X (2018) J Org Chem 83:4618
222. Han Z, Wang Z, Zhang X, Ding K (2009) Angew Chem Int Ed 48:5345
223. Welch WM, Kraska AR, Sarges R, Koe BK (1984) J Med Chem 27:1508
224. Qu B, Samankumara LP, Ma S, Fandrick KR, Desrosiers JN, Rodriguez S, Li Z, Haddad N,
Han ZS, McKellop K, Pennino S, Grinberg N, Gonnella NC, Song JJ, Senanayake CH (2014)
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225. Hou CJ, Wang YH, Zheng Z, Xu J, Hu XP (2012) Org Lett 14:3554
226. Li Q, Hou CJ, Liu XN, Huang DZ, Liu YJ, Yanga RF, Hu XP (2015) RSC Adv 5:13702
227. Bishop MJ, McNutt RW (1995) Bioorg Med Chem Lett 5:1311
228. Spencer CM, Foulds D, Peters DH (1993) Drugs 46:1055
229. Sakurai S, Ogawa N, Suzuki T, Kato K, Ohashi T, Yasuda S, Kato H, Ito Y (1996) Chem
Pharm Bull 44:765
230. Tulshian D, Ho GD, Silverman L, Matasi JJ, McLeod RL, Hey JA, Chapman RW,
Bercovici A, Cuss FM, WO 01/07050 A1 (Schering-Plough)
231. Jolidon S, Narquizian R, Pinard E. WO 2008/022938 A1 (Hoffman-LaRoche)
232. Ducray P, Cavaliero T, Lorhmann M, Bouvier J WO 2008/062006 A1 (Novartis)
202
J. Margalef et al.
194. Li S, Xiao T, Li D, Zhang X (2015) Org Lett 17:3782
195. Xie JH, Zhu SF, Zhou QL (2012) Chem Soc Rev 41:4126
196. Maire P, Deblon S, Breher F, Geier J, Böhler C, Rüegger H, Schönberg H, Grützmacher H
(2004) Chem Eur J 10:4198
197. Giacomina F, Meetsma A, Panella L, Lefort L, de Vries AHM, de Vries JG (2007) Angew
Chem Int Ed 46:1497
198. Enthaler S, Erre G, Junge K, Schröder K, Addis D, Michalik D, Hapke M, Redkin D, Beller M
(2008) Eur J Org Chem:3352
199. Erre G, Enthaler S, Junge K, Addis D, Beller M (2009) Adv Synth Catal 351:1437
200. Hou G, Li W, Ma M, Zhang X, Zhang X (2010) J Am Chem Soc 132:12844
201. Busscher GF, Lefort L, Cremers JGO, Mottinelli M, Wiertz RW, de Lange B, Okamura Y,
Yusa Y, Matsumura K, Shimizu H, de Vries JG, de Vries AHM (2010) Tetrahedron Asymmetry 21:1709
202. Han Z, Guan YQ, Liu G, Wang R, Yin X, Zhao Q, Cong H, Dong XQ, Zhang X (2018) Org
Lett 20:6349
203. Patureau FW, Worch C, Siegler MA, Spek AL, Bolm C, Reek JNH (2012) Adv Synth Catal
354:59
204. Margalef J, Pàmies O, Diéguez M (2017) Chem Eur J 23:813
205. Cabré A, Verdaguer X, Riera A (2019) Adv Synth Catal 361:4196
206. Cabré A, Romagnoli E, Martínez-Balart P, Verdaguer X, Riera A (2019) Org Lett 21:9709
207. Lazarevski G, Kobrehel G, Metelko B, Duddeck H (1996) J Antibiot 49:1066
208. Nicholas GM, Molinski TF (2000) Tetrahedron 56:2921
209. Davies HML, Ni A (2006) Chem Commun:3110
210. Harris RN, Stabler RS, Repke DB, Kress JM, Walker KA, Martin RS, Brothers JM, Ilnicka M,
Lee SW, Mirzadegan T (2010) Bioorg Med Chem Lett 20:3436
211. Ramesh P, Suman D (2018) Synthesis 50:211
212. Fleury-Brégeot N, de la Fuente V, Castillón S (2010) ChemCatChem 2:1346
213. Xie JH, Zhu SF, Zhou QL (2011) Chem Rev 111:1713
214. James BR (1997) Catal Today 37:209
215. Blaser HU, Buser HP, Loers K, Hanreich R, Jalett HP, Jelsch E, Pugin B, Schneider HD,
Spindler F, Wagmann A (1999) Chimia 53:275
216. Xiao D, Zhang X (2001) Angew Chem Int Ed 40:3425
217. Mršić N, Panella L, Ijpeij EJ, Minnaard AJ, Feringa BL, De Vries JG (2011) ChemCatChem
3:1139
218. Baeza A, Pfaltz A (2010) Chem Eur J 16:4003
219. Schramm Y, Barrios-Landeros F, Pfaltz A (2013) Chem Sci 4:2760
220. Salomó E, Gallen A, Sciortino G, Ujaque G, Grabulosa A, Lledós A, Riera A, Verdaguer X
(2018) J Am Chem Soc 140:16967
221. Salomó E, Rojo P, Hernández-Lladó P, Riera A, Verdaguer X (2018) J Org Chem 83:4618
222. Han Z, Wang Z, Zhang X, Ding K (2009) Angew Chem Int Ed 48:5345
223. Welch WM, Kraska AR, Sarges R, Koe BK (1984) J Med Chem 27:1508
224. Qu B, Samankumara LP, Ma S, Fandrick KR, Desrosiers JN, Rodriguez S, Li Z, Haddad N,
Han ZS, McKellop K, Pennino S, Grinberg N, Gonnella NC, Song JJ, Senanayake CH (2014)
Angew Chem Int Ed 53:14428
225. Hou CJ, Wang YH, Zheng Z, Xu J, Hu XP (2012) Org Lett 14:3554
226. Li Q, Hou CJ, Liu XN, Huang DZ, Liu YJ, Yanga RF, Hu XP (2015) RSC Adv 5:13702
227. Bishop MJ, McNutt RW (1995) Bioorg Med Chem Lett 5:1311
228. Spencer CM, Foulds D, Peters DH (1993) Drugs 46:1055
229. Sakurai S, Ogawa N, Suzuki T, Kato K, Ohashi T, Yasuda S, Kato H, Ito Y (1996) Chem
Pharm Bull 44:765
230. Tulshian D, Ho GD, Silverman L, Matasi JJ, McLeod RL, Hey JA, Chapman RW,
Bercovici A, Cuss FM, WO 01/07050 A1 (Schering-Plough)
231. Jolidon S, Narquizian R, Pinard E. WO 2008/022938 A1 (Hoffman-LaRoche)
232. Ducray P, Cavaliero T, Lorhmann M, Bouvier J WO 2008/062006 A1 (Novartis)
202
J. Margalef et al.
