316
249. Sharma A, Vacchani D, Van der Eycken E (2013) Developments in Direct C–H Arylation of
(Hetero)Arenes under Microwave Irradiation. Chem Eur J 19:1158
250. Gupta AK, Singh N, Singh KN (2013) Microwave Assisted Organic Synthesis: Cross
Coupling and Multicomponent Reactions. Curr Org Chem 17:474
251. Besson T, Fruit C (2016) Recent Developments in Microwave-Assisted Metal-Catalyzed
C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications.
Synthesis 48:3879
252. Baber RA, Bedford RB, Betham M, Blake ME, Coles SJ, Haddow MF, Hursthouse MB,
Orpen AG, Pilarski LT, Pringle PG, Wingad RL, (2006) Chiral palladium bis(phosphite)
PCP-pincer complexes via ligand C-H activation. Chem Commun 37:3880
253. Sridharan V, Martín MA, Menéndez JC (2009) Acid-Free Synthesis of Carbazoles and
Carbazolequinones by Intramolecular Pd‐Catalyzed, Microwave-Assisted Oxidative Biaryl
Coupling Reactions - Efficient Syntheses of Murrayafoline A, 2-Methoxy-3-methylcarbazole,
and Glycozolidine. Eur J Org Chem 27:4614
254. Mahindra A, Bagra N, Jain R (2013) Palladium-Catalyzed Regioselective C-5 Arylation of
Protected l-Histidine: Microwave-Assisted C–H Activation Adjacent to Donor Arm. J Org
Chem 78:10954
255. Choi S J, Kuwabara J, Kanbara T (2013) Microwave-Assisted Polycondensation via Direct
Arylation of 3,4-Ethylenedioxythiophene with 9,9-Dioctyl-2,7-dibromofluorene. ACS
Sustainable Chem Eng 1:878
256. Kokornaczyk A, Schepmann D, Yamaguchi J, Itamib K, Wünsch B (2016) Microwaveassisted regioselective direct C–H arylation of thiazole derivatives leading to increased σ1
receptor affinity. Med Chem Commun 7:327
257. Baladi T, Granzhan A, Piguel S (2016) Microwave‐Assisted C‐2 Direct Alk enylation of
Imidazo[4,5‐b]pyr idines: Access to Fluorescent Purine Isosteres with Remarkably Large
Stokes Shifts. Eur J Org Chem 2016:2421
258. Harari M, Couly F, Fruit C, Besson T (2016) Pd-Catalyzed and Copper Assisted Regioselective
Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.
Org Lett 18:3282
259. Godeau J, Harari M, Laclef S, Deau E, Fruit C, Besson T (2015) Cu/Pd‐Catalyzed C‐2–H
Arylation of Quinazolin‐4(3H)‐ones with (Hetero)aryl Halides. Eur J Org Chem 35: 7705
260. Li S, Wan P, Ai J, Sheng R, Hu Y, Hu Y (2017) Palladium-Catalyzed, Silver-Assisted Direct
C-5-H Arylation of 3‐Substituted 1,2,4‐Oxadiazoles under Microwave Irradiation. Adv Synth
Catal 359:772
261. Khlebnikov V, Heckenroth M, Müller-Bunz H, Albrecht M (2013) Platinum(ii) and
platinum(iv) complexes stabilized by abnormal/mesoionic C4-bound dicarbenes. Dalton
Trans 42:4197
262. Diness F, Begtrup M (2014) Sequential Direct SNAr Reactions of Pentafluorobenzenes with
Azole or Indole Derivatives. Org Lett 16:3130
263. Mfuh AM, Larionov OV (2015) Heterocyclic N-Oxides - An Emerging Class of Therapeutic
Agents. Curr Med Chem 22:2819
264. Stephens DE, Lakey-Beita J, Atesin AC, Ateşin TA, Chavez G, Arman HD, Larionov OV
(2015) Palladium-Catalyzed C8-Selective C–H Arylation of Quinoline N-Oxides: Insights
into the Electronic, Steric, and Solvation Effects on the Site Selectivity by Mechanistic and
DFT Computational Studies. ACS Catal 5:167
265. Stephens DE, Lakey-Beita J, Chavez G, Ilie C, Arman HD, Larionov OV (2015) Experimental
and mechanistic analysis of the palladium-catalyzed oxidative C8-selective C-H homocoupling of quinoline N-oxides. Chem Commun 51:9507
266. Vachhani DD, Sharma A, Van der Eycken E (2013) Copper-catalyzed direct secondary and
tertiary C-H alkylation of azoles through a heteroarene-amine-aldehyde/ketone coupling
reaction. Angew Chem Int Ed 52:2547
D. S. Deshmukh et al.
249. Sharma A, Vacchani D, Van der Eycken E (2013) Developments in Direct C–H Arylation of
(Hetero)Arenes under Microwave Irradiation. Chem Eur J 19:1158
250. Gupta AK, Singh N, Singh KN (2013) Microwave Assisted Organic Synthesis: Cross
Coupling and Multicomponent Reactions. Curr Org Chem 17:474
251. Besson T, Fruit C (2016) Recent Developments in Microwave-Assisted Metal-Catalyzed
C–H Functionalization of Heteroarenes for Medicinal Chemistry and Material Applications.
Synthesis 48:3879
252. Baber RA, Bedford RB, Betham M, Blake ME, Coles SJ, Haddow MF, Hursthouse MB,
Orpen AG, Pilarski LT, Pringle PG, Wingad RL, (2006) Chiral palladium bis(phosphite)
PCP-pincer complexes via ligand C-H activation. Chem Commun 37:3880
253. Sridharan V, Martín MA, Menéndez JC (2009) Acid-Free Synthesis of Carbazoles and
Carbazolequinones by Intramolecular Pd‐Catalyzed, Microwave-Assisted Oxidative Biaryl
Coupling Reactions - Efficient Syntheses of Murrayafoline A, 2-Methoxy-3-methylcarbazole,
and Glycozolidine. Eur J Org Chem 27:4614
254. Mahindra A, Bagra N, Jain R (2013) Palladium-Catalyzed Regioselective C-5 Arylation of
Protected l-Histidine: Microwave-Assisted C–H Activation Adjacent to Donor Arm. J Org
Chem 78:10954
255. Choi S J, Kuwabara J, Kanbara T (2013) Microwave-Assisted Polycondensation via Direct
Arylation of 3,4-Ethylenedioxythiophene with 9,9-Dioctyl-2,7-dibromofluorene. ACS
Sustainable Chem Eng 1:878
256. Kokornaczyk A, Schepmann D, Yamaguchi J, Itamib K, Wünsch B (2016) Microwaveassisted regioselective direct C–H arylation of thiazole derivatives leading to increased σ1
receptor affinity. Med Chem Commun 7:327
257. Baladi T, Granzhan A, Piguel S (2016) Microwave‐Assisted C‐2 Direct Alk enylation of
Imidazo[4,5‐b]pyr idines: Access to Fluorescent Purine Isosteres with Remarkably Large
Stokes Shifts. Eur J Org Chem 2016:2421
258. Harari M, Couly F, Fruit C, Besson T (2016) Pd-Catalyzed and Copper Assisted Regioselective
Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.
Org Lett 18:3282
259. Godeau J, Harari M, Laclef S, Deau E, Fruit C, Besson T (2015) Cu/Pd‐Catalyzed C‐2–H
Arylation of Quinazolin‐4(3H)‐ones with (Hetero)aryl Halides. Eur J Org Chem 35: 7705
260. Li S, Wan P, Ai J, Sheng R, Hu Y, Hu Y (2017) Palladium-Catalyzed, Silver-Assisted Direct
C-5-H Arylation of 3‐Substituted 1,2,4‐Oxadiazoles under Microwave Irradiation. Adv Synth
Catal 359:772
261. Khlebnikov V, Heckenroth M, Müller-Bunz H, Albrecht M (2013) Platinum(ii) and
platinum(iv) complexes stabilized by abnormal/mesoionic C4-bound dicarbenes. Dalton
Trans 42:4197
262. Diness F, Begtrup M (2014) Sequential Direct SNAr Reactions of Pentafluorobenzenes with
Azole or Indole Derivatives. Org Lett 16:3130
263. Mfuh AM, Larionov OV (2015) Heterocyclic N-Oxides - An Emerging Class of Therapeutic
Agents. Curr Med Chem 22:2819
264. Stephens DE, Lakey-Beita J, Atesin AC, Ateşin TA, Chavez G, Arman HD, Larionov OV
(2015) Palladium-Catalyzed C8-Selective C–H Arylation of Quinoline N-Oxides: Insights
into the Electronic, Steric, and Solvation Effects on the Site Selectivity by Mechanistic and
DFT Computational Studies. ACS Catal 5:167
265. Stephens DE, Lakey-Beita J, Chavez G, Ilie C, Arman HD, Larionov OV (2015) Experimental
and mechanistic analysis of the palladium-catalyzed oxidative C8-selective C-H homocoupling of quinoline N-oxides. Chem Commun 51:9507
266. Vachhani DD, Sharma A, Van der Eycken E (2013) Copper-catalyzed direct secondary and
tertiary C-H alkylation of azoles through a heteroarene-amine-aldehyde/ketone coupling
reaction. Angew Chem Int Ed 52:2547
D. S. Deshmukh et al.