References
91
103. Conde S, Corral C, Madronero R (1974) Synthesis of 1H-1,2,4-Triazoles via Nitrillium Salts.
Synthesis (Stuttg) 28–29
104. Wang L-Y, Tsai HJ, Lin H-Y, Kaneko K, Cheng F-Y, Shih H-S, Wong FF, Huang J-J (2014)
One-flask synthesis of 1,3,5-Trisubstituted 1,2,4-Triazoles from Nitriles and Hydrazonoyl
chlorides via 1,3-dipolar cycloaddition. RSC Adv 4:14215–14220
105. Huisgen R, Grashey R, Seidel M, Knupfer H, Schmidt R (1962) 1.3-Dipolare Additionen, III.
Umsetzungen des Diphenylnitrilimins mit Carbonyl und Thiocarbonyl-Verbindungen. Justus
Liebigs Ann Chem 658:169–180
106. Elmoghayar MRH, Elnagdi MH, Ibrahim MKA, Sallam MMM (1977) Reactions
with Carbo(heterylhydrazonoyl) Halides. I. Chemistry of Carbo(3-phenylpyrazol-5-ylhydrazonoyl) Chlorides. Helv Chim Acta 60:2171–2176
107. Schoder F, Plaia U, Metzner R, Sperber W, Beck W, Fehlhammer WP (2010) [3 + 2]
Cycloadditions of metallo nitrile ylides and metallo nitrile imines with metal carbonyl,
thiocarbonyl, and isocyanide complexes: heterodimetallic systems with bridging heterocycles.
Zeitschrift für Anorg und Allg Chemie 636:700–709
108. Feddouli A, Itto MYA, Hasnaoui A, Villemin D, Jaffrès P-A, Santos JS-DO, Riahi A, Huet F,
Daran J-C (2004) One pot diastereoselective synthesis of new chiral spiro-1,3,4-Thiadiazoles
and 1,4,2-oxathiazoles from (1R)-Thiocamphor. J Heterocycl Chem 41:731–735
109. Utecht G, Sioma J, Jasinkski M, Mloston G (2017) Expected and unexpected results in
reactions of fluorinated nitrile imines with (Cyclo)aliphatic thioketones. J Fluor Chem
201:68–75
110. Katada T, Eguchi S, Sasaki T (1984) Thermal cycloaddition reactions of thiocarbonyl
compounds. Part 2. 1,3-dipolar cycloaddition reactions of adamantanethione with nitrile
oxides, nitrilimines, and diazoalkanes. J Chem Soc Perkin Trans 1 2641
111. Grubert L, Pätzel M, Jugelt W, Riemer B, Liebscher J (1994) Reaktionen von 1,3-Dipolen
mit Heterocyclen, 9. Umsetzungen von Nitriliminen mit Pyrazinen, Pyrimidinen und 1HPyrimidinthionen. Liebigs Ann der Chemie 1994:1005–1011
112. Büchel T, Prewo R, Bieri JH, Heimgartner H (1984) 1,3-dipolare cycloadditionen von
nitrilium-betainen mit 4,4-Dimethyl-2-phenyl-2-thiazolin-5-thion. Helv Chim Acta 67:534–
549
113. Barriga S, Fuertes P, Marcos CF, Miguel D, Rakitin OA, Rees CW, Torroba T (2001) Synthesis
of thiadiazole, dithietane, and imine derivatives of the [1,2]Dithiolo[1,4]thiazine ring system.
J Org Chem 66:5766–5771
114. Bohrisch J, Pätzel M, Grubert L, Liebscher J (1993) Synthesis of S, N-heterocycles from
N-thioacyllactamimines. Phosphorus, Sulfur Silicon Relat Elem 84:253–256
115. Abouricha S, Rakib EM, Benchat N, Alaoui M, Allouchi H, El Bali B (2005) Facile synthesis of
new spirothiadiazolopyridazines by 1,3-dipolar cycloaddition. Synth Commun 35:2213–2221
116. Bonini BF, Mazzanti G, Sarti S, Zanirato P, Maccagnani G (1981) Silyl thioketones and
silylated thiirans. J Chem Soc Chem Commun 822
117. Greig DJ, McPherson M, Paton RM, Crosby J (1985) Cycloaddition reactions of 1,4,2Dithiazole-5-thiones. J Chem Soc Perkin Trans 1:1205
118. Dickoré K, Wegler R (1966) Formation of 1,3,4-Thiadiazoles and 1,4,2-Oxathiazoles from
thioketenes. Angew Chemie Int Ed Engl 5:970
119. Linden A, Awad EMAH, Heimgartner H (1999) A rhodanine derivative and its cycloadduct
with diphenyl nitrile Imine. Acta Crystallogr Sect C: Cryst Struct Commun 55:1877–1881
120. Friedrich K, Zamkanei M (1979) Cycloadditionen von cyanthioformamiden mit 1,3-Dipolen.
Chem Ber 112:1873–1878
121. Huisgen R (1963) 1,3-dipolar cycloadditions. past and future. Angew Chemie Int Ed Engl
2:565–598
122. Wustrow DJ, Belliotti TR, Capiris T, Kneen CO, Bryans JS, Field MJ, Williams D, El-Kattan
A, Buchholz L, Kinsora JJ, Lotarski SM, Vartanian MG, Taylor CP, Donevan SD, Thorpe
AJ, Schwarz JB (2009) Oxadiazolone bioisosteres of pregabalin and gabapentin. Bioorg Med
Chem Lett 19:247–250
91
103. Conde S, Corral C, Madronero R (1974) Synthesis of 1H-1,2,4-Triazoles via Nitrillium Salts.
Synthesis (Stuttg) 28–29
104. Wang L-Y, Tsai HJ, Lin H-Y, Kaneko K, Cheng F-Y, Shih H-S, Wong FF, Huang J-J (2014)
One-flask synthesis of 1,3,5-Trisubstituted 1,2,4-Triazoles from Nitriles and Hydrazonoyl
chlorides via 1,3-dipolar cycloaddition. RSC Adv 4:14215–14220
105. Huisgen R, Grashey R, Seidel M, Knupfer H, Schmidt R (1962) 1.3-Dipolare Additionen, III.
Umsetzungen des Diphenylnitrilimins mit Carbonyl und Thiocarbonyl-Verbindungen. Justus
Liebigs Ann Chem 658:169–180
106. Elmoghayar MRH, Elnagdi MH, Ibrahim MKA, Sallam MMM (1977) Reactions
with Carbo(heterylhydrazonoyl) Halides. I. Chemistry of Carbo(3-phenylpyrazol-5-ylhydrazonoyl) Chlorides. Helv Chim Acta 60:2171–2176
107. Schoder F, Plaia U, Metzner R, Sperber W, Beck W, Fehlhammer WP (2010) [3 + 2]
Cycloadditions of metallo nitrile ylides and metallo nitrile imines with metal carbonyl,
thiocarbonyl, and isocyanide complexes: heterodimetallic systems with bridging heterocycles.
Zeitschrift für Anorg und Allg Chemie 636:700–709
108. Feddouli A, Itto MYA, Hasnaoui A, Villemin D, Jaffrès P-A, Santos JS-DO, Riahi A, Huet F,
Daran J-C (2004) One pot diastereoselective synthesis of new chiral spiro-1,3,4-Thiadiazoles
and 1,4,2-oxathiazoles from (1R)-Thiocamphor. J Heterocycl Chem 41:731–735
109. Utecht G, Sioma J, Jasinkski M, Mloston G (2017) Expected and unexpected results in
reactions of fluorinated nitrile imines with (Cyclo)aliphatic thioketones. J Fluor Chem
201:68–75
110. Katada T, Eguchi S, Sasaki T (1984) Thermal cycloaddition reactions of thiocarbonyl
compounds. Part 2. 1,3-dipolar cycloaddition reactions of adamantanethione with nitrile
oxides, nitrilimines, and diazoalkanes. J Chem Soc Perkin Trans 1 2641
111. Grubert L, Pätzel M, Jugelt W, Riemer B, Liebscher J (1994) Reaktionen von 1,3-Dipolen
mit Heterocyclen, 9. Umsetzungen von Nitriliminen mit Pyrazinen, Pyrimidinen und 1HPyrimidinthionen. Liebigs Ann der Chemie 1994:1005–1011
112. Büchel T, Prewo R, Bieri JH, Heimgartner H (1984) 1,3-dipolare cycloadditionen von
nitrilium-betainen mit 4,4-Dimethyl-2-phenyl-2-thiazolin-5-thion. Helv Chim Acta 67:534–
549
113. Barriga S, Fuertes P, Marcos CF, Miguel D, Rakitin OA, Rees CW, Torroba T (2001) Synthesis
of thiadiazole, dithietane, and imine derivatives of the [1,2]Dithiolo[1,4]thiazine ring system.
J Org Chem 66:5766–5771
114. Bohrisch J, Pätzel M, Grubert L, Liebscher J (1993) Synthesis of S, N-heterocycles from
N-thioacyllactamimines. Phosphorus, Sulfur Silicon Relat Elem 84:253–256
115. Abouricha S, Rakib EM, Benchat N, Alaoui M, Allouchi H, El Bali B (2005) Facile synthesis of
new spirothiadiazolopyridazines by 1,3-dipolar cycloaddition. Synth Commun 35:2213–2221
116. Bonini BF, Mazzanti G, Sarti S, Zanirato P, Maccagnani G (1981) Silyl thioketones and
silylated thiirans. J Chem Soc Chem Commun 822
117. Greig DJ, McPherson M, Paton RM, Crosby J (1985) Cycloaddition reactions of 1,4,2Dithiazole-5-thiones. J Chem Soc Perkin Trans 1:1205
118. Dickoré K, Wegler R (1966) Formation of 1,3,4-Thiadiazoles and 1,4,2-Oxathiazoles from
thioketenes. Angew Chemie Int Ed Engl 5:970
119. Linden A, Awad EMAH, Heimgartner H (1999) A rhodanine derivative and its cycloadduct
with diphenyl nitrile Imine. Acta Crystallogr Sect C: Cryst Struct Commun 55:1877–1881
120. Friedrich K, Zamkanei M (1979) Cycloadditionen von cyanthioformamiden mit 1,3-Dipolen.
Chem Ber 112:1873–1878
121. Huisgen R (1963) 1,3-dipolar cycloadditions. past and future. Angew Chemie Int Ed Engl
2:565–598
122. Wustrow DJ, Belliotti TR, Capiris T, Kneen CO, Bryans JS, Field MJ, Williams D, El-Kattan
A, Buchholz L, Kinsora JJ, Lotarski SM, Vartanian MG, Taylor CP, Donevan SD, Thorpe
AJ, Schwarz JB (2009) Oxadiazolone bioisosteres of pregabalin and gabapentin. Bioorg Med
Chem Lett 19:247–250