96
3 The Reactivity of Nitrile Imines
209. Jayashankar B, Lokanatha Rai KM, Baskaran N, Sathish HS (2009) Synthesis and
pharmacological evaluation of 1,3,4-oxadiazole bearing Bis(heterocycle) derivatives as
anti-inflammatory and analgesic agents. Eur J Med Chem 44:3898–3902
210. Gaonkar SL, Rai KML, Prabhuswamy B (2006) Synthesis and antimicrobial studies of a new
series of 2-{4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl}-5-substituted-1,3,4-oxadiazoles. Eur J
Med Chem 41:841–846
211. Gibson MS (1962) Hydrazones—III: intramolecular 1,3-dipolar additions involving nitroand carbonyl groups. Tetrahedron 18:1377–1380
212. Gladstone WAF, Aylward JB, Norman ROC (1969) Reactions of lead tetra-acetate. Part XVIII.
Oxidation of aldehyde hydrazones: a new method for the generation of nitrilimines. J Chem
Soc C Org 2587
213. Huisgen R, Sauer J, Sturm HJ, Markgraf JH (1960) Ringöffnungen der Azole, II. Die bildung
von 1.3.4-Oxdiazolen bei der Acylierung 5-substituierter Tetrazole. Chem Ber 93:2106–2124
214. Adelstein GW (1973) Antiarrhythmic agents. Synthesis and biological activity of some
tetrazole and oxadiazole analogs of 4-Dialkylamino-2,2-Diarylbutyramides. J Med Chem
16:309–312
215. Wamhoff H, Zahran M (1987) Dihalogentriphenylphosphoranes in heterocyclic synthesis;
15.1 A simple one-pot-procedure for the generation of nitrilimines with the aid of
dihalogentriphenyl-phosphoranes: 1,3-Dipolar cycloadditions and 1,5-electrocyclizations.
Synthesis (Stuttg) 876–879
216. Huisgen R, Sauer J, Seidel M (1960) Ringöffnungen der Azole, IV. Die synthese von 1.2.4Triazolen aus 5-substituierten tetrazolen und Carbonsäure-imidchloriden. Chem Ber 93:2885–
2891
217. Konnecke A, Lippmann E (1977) N-Hetaryltetrazoles—I. Tetrazolyltetrazolo/1,5a/pyrimidines, intermediates in the formation of s-Triazolo/4,3-c/tetrazolo/1,5-a/pyrimidines.
Tetrahedron Lett 18:2187–2188
218. Huisgen R, Sturm HJ, Seidel M (1961) Ringöffnungen der Azole, V. Weitere Reaktionen der
Tetrazole mit elektrophilen Agenzien. Chem Ber 94:1555–1562
219. Maas G, Gümbel H, Weise G, Regitz M (1985) Untersuchungen an Diazoverbindungen und
Aziden, 58. Dikation-ether, 5. Formamidinium-substituierte Diazophosphoryl-Verbindungen:
Synthese, Eigenschaften und Reaktionen zu Tetrazolen. Chem Ber 118:2105–2117
220. Moody CJ, Rees CW, Young RG (1991) Synthesis of 3-phenylpyrazoles from 2-alkenyl-5phenytetrazoles. J Chem Soc Perkin Trans 1:329
221. Granier M, Baceiredo A, Nieger M, Bertrand G (1990) An N-phosphino C-thiophosphinoyi
nitrilimine as a formal 1,4 dipole: synthesis of 1,2,3λ5-Diaza- and 1,2,4,3λ5Triazaphosphinines. Angew Chemie Int Ed Engl 29:1123–1125
222. Huisgen R, Weberndörfer V (1967) 1.3-Dipolare cycloadditionen, XXVI. Intramolekulare
Stabilisierung bei einem N-Trinitrophenylnitrilimin. Chem Ber 100:71–78
223. Barnish IT, Gibson MS (1968) Rearrangement during dehydrobromination of hydrazidic
bromides derived from o-Nitrophenylhydrazine, and a comment on the nitration of pdibromobenzene. J Chem Soc C Org 8–11
224. Könnecke A, Lepom P, Lippmann E (1978) Synthesis and thermolysis of 5-Aryl-2-(2,4Dinitrophenyl) tetrazoles. Zeitschrift für Chemie 18:214–215
225. König W, Geiger R (1970) Eine neue Methode zur Synthese von Peptiden: Aktivierung der
Carboxylgruppe mit Dicyclohexylcarbodiimid unter Zusatz von 1-Hydroxy-benzotriazolen.
Chem Ber 103:788–798
226. Konnecke A, Dorre R, Lippmann E (1978) N-Hetaryltetrazoles-III, competitive
intramolecular 1, x-Dipolar Cyclizations of thermally produced nitilimines. Tetrahedron Lett
19:2071–2074
227. Nunes CM, Reva I, Rosado MTS, Fausto R (2015) The quest for carbenic nitrile imines:
experimental and computational characterization of C-Amino Nitrile Imine. Eur J Org Chem
7484–7493
228. Bégué D, Wentrup C (2014) Carbenic nitrile imines: properties and reactivity. J Org Chem
79:1418–1426
3 The Reactivity of Nitrile Imines
209. Jayashankar B, Lokanatha Rai KM, Baskaran N, Sathish HS (2009) Synthesis and
pharmacological evaluation of 1,3,4-oxadiazole bearing Bis(heterocycle) derivatives as
anti-inflammatory and analgesic agents. Eur J Med Chem 44:3898–3902
210. Gaonkar SL, Rai KML, Prabhuswamy B (2006) Synthesis and antimicrobial studies of a new
series of 2-{4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl}-5-substituted-1,3,4-oxadiazoles. Eur J
Med Chem 41:841–846
211. Gibson MS (1962) Hydrazones—III: intramolecular 1,3-dipolar additions involving nitroand carbonyl groups. Tetrahedron 18:1377–1380
212. Gladstone WAF, Aylward JB, Norman ROC (1969) Reactions of lead tetra-acetate. Part XVIII.
Oxidation of aldehyde hydrazones: a new method for the generation of nitrilimines. J Chem
Soc C Org 2587
213. Huisgen R, Sauer J, Sturm HJ, Markgraf JH (1960) Ringöffnungen der Azole, II. Die bildung
von 1.3.4-Oxdiazolen bei der Acylierung 5-substituierter Tetrazole. Chem Ber 93:2106–2124
214. Adelstein GW (1973) Antiarrhythmic agents. Synthesis and biological activity of some
tetrazole and oxadiazole analogs of 4-Dialkylamino-2,2-Diarylbutyramides. J Med Chem
16:309–312
215. Wamhoff H, Zahran M (1987) Dihalogentriphenylphosphoranes in heterocyclic synthesis;
15.1 A simple one-pot-procedure for the generation of nitrilimines with the aid of
dihalogentriphenyl-phosphoranes: 1,3-Dipolar cycloadditions and 1,5-electrocyclizations.
Synthesis (Stuttg) 876–879
216. Huisgen R, Sauer J, Seidel M (1960) Ringöffnungen der Azole, IV. Die synthese von 1.2.4Triazolen aus 5-substituierten tetrazolen und Carbonsäure-imidchloriden. Chem Ber 93:2885–
2891
217. Konnecke A, Lippmann E (1977) N-Hetaryltetrazoles—I. Tetrazolyltetrazolo/1,5a/pyrimidines, intermediates in the formation of s-Triazolo/4,3-c/tetrazolo/1,5-a/pyrimidines.
Tetrahedron Lett 18:2187–2188
218. Huisgen R, Sturm HJ, Seidel M (1961) Ringöffnungen der Azole, V. Weitere Reaktionen der
Tetrazole mit elektrophilen Agenzien. Chem Ber 94:1555–1562
219. Maas G, Gümbel H, Weise G, Regitz M (1985) Untersuchungen an Diazoverbindungen und
Aziden, 58. Dikation-ether, 5. Formamidinium-substituierte Diazophosphoryl-Verbindungen:
Synthese, Eigenschaften und Reaktionen zu Tetrazolen. Chem Ber 118:2105–2117
220. Moody CJ, Rees CW, Young RG (1991) Synthesis of 3-phenylpyrazoles from 2-alkenyl-5phenytetrazoles. J Chem Soc Perkin Trans 1:329
221. Granier M, Baceiredo A, Nieger M, Bertrand G (1990) An N-phosphino C-thiophosphinoyi
nitrilimine as a formal 1,4 dipole: synthesis of 1,2,3λ5-Diaza- and 1,2,4,3λ5Triazaphosphinines. Angew Chemie Int Ed Engl 29:1123–1125
222. Huisgen R, Weberndörfer V (1967) 1.3-Dipolare cycloadditionen, XXVI. Intramolekulare
Stabilisierung bei einem N-Trinitrophenylnitrilimin. Chem Ber 100:71–78
223. Barnish IT, Gibson MS (1968) Rearrangement during dehydrobromination of hydrazidic
bromides derived from o-Nitrophenylhydrazine, and a comment on the nitration of pdibromobenzene. J Chem Soc C Org 8–11
224. Könnecke A, Lepom P, Lippmann E (1978) Synthesis and thermolysis of 5-Aryl-2-(2,4Dinitrophenyl) tetrazoles. Zeitschrift für Chemie 18:214–215
225. König W, Geiger R (1970) Eine neue Methode zur Synthese von Peptiden: Aktivierung der
Carboxylgruppe mit Dicyclohexylcarbodiimid unter Zusatz von 1-Hydroxy-benzotriazolen.
Chem Ber 103:788–798
226. Konnecke A, Dorre R, Lippmann E (1978) N-Hetaryltetrazoles-III, competitive
intramolecular 1, x-Dipolar Cyclizations of thermally produced nitilimines. Tetrahedron Lett
19:2071–2074
227. Nunes CM, Reva I, Rosado MTS, Fausto R (2015) The quest for carbenic nitrile imines:
experimental and computational characterization of C-Amino Nitrile Imine. Eur J Org Chem
7484–7493
228. Bégué D, Wentrup C (2014) Carbenic nitrile imines: properties and reactivity. J Org Chem
79:1418–1426