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imines by the sulphide function. J Chem Soc, Perkin Trans 1:2535–2539
161. Meier Hansruedi, Heinzelmann Willy, Heimgartner H (1980) Inter- and intramolecular
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162. Zhao S, Dai J, Hu M, Liu C, Meng R, Liu X, Wang C, Luo T (2016) Photo-induced coupling
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163. Herner A, Marjanovic J, Lewandowski TM, Marin V, Patterson M, Miesbauer L, Ready D,
Williams J, Vasudevan A, Lin Q (2016) 2-Aryl-5-carboxytetrazole as a new photoaffinity
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164. Heiler C, Offenloch JT, Blasco E, Barner-Kowollik C (2017) Photochemically induced folding
of single chain polymer nanoparticles in water. ACS Macro Lett 6:56–61
165. Konrad W, Fengler C, Putwa S, Barner-Kowollik C (2019) Protection-group-free synthesis
of sequence-defined macromolecules via precision λ-orthogonal photochemistry. Angew
Chemie Int Ed 58:7133–7137
93
144. Aylward JB, Scott FL (1970) Synthesis and properties of alkyl hydrazonates. J Chem Soc C
Org 968
145. Shawali AS, Hassaneen HM (1972) Synthesis and rearrangement of hydrazones of aryl
benzoates. Tetrahedron Lett 13:1299–1300
146. Shawali AS, Sami M, Sherif SM, Párkányi C (1980) Synthesis of some derivatives
of imidazo[1,2-a]pyridine, Pyrazolo[1,5-b]imidazole, and 4-(3H)Quinazolinone from αKetohydrazidoyl bromides. J Heterocycl Chem 17:877–880
147. El-Abadelah MM, Nazer MZ, El-Abadlah NS, Meier H (1997) Synthesis of
methyl 4-Amino-1-aryl-1,4,5,6-Tetrahydro-6-oxo-1,2,4-Triazine-3-carboxylates. J für Prakt
Chemie/Chemiker-Zeitung 339:90–91
148. Abu Thaher BA, Zahra JA, El-Abadelah MM (2002) Facile synthesis of model 1,4-dihydro1H-1,3,4-benzotriazepin-5-ones. J Heterocycl Chem 39:901–904
149. Abu Thaher B, Zahra JA, El-Abadelah MM, Otto H-H (2004) On the synthesis of 3Acetyl-1-aryl-1,4,5,6-tetrahydro-1H-1,2,4-triazepin-7-ones by reaction of nitrilimines with
3-aminopropanoic acid. Monatsh Chem 135:435–439
150. Hindawi NI, Zahra JA, El-Abadelah MM, Abu Thaher BA, Zeller K-P (2006) Facile synthesis
of dihydro-1,2,4-benzotriazepin-5-ones. Monatshefte für Chemie. Chem Mon 137:1349–1355
151. Dalloul HM (2008) Synthesis of nitrogen-containing dispiroheterocycles (1) using
nitrilimines. ARKIVOC 14:243–247
152. Dalloul HMM (2011) Synthesis of spiroheterocycles containing thiadiazole thiadiazine and
triazine moieties from nitrilimines. Phosphorus, Sulfur Silicon Relat Elem 186:1876–1884
153. Mustafa MS, El-Abadelah MM, Mubarak MS, Chibueze I, Shao D, Agu RU (2011) Synthesis
and fluorogenic properties of some 1-(Coumarin-7-yl)-4,5-dihydro-1,2,4-triazin-6(1H)-ones.
Int J Chem 3:89
154. Dalloul HMM (2009) Heterocyclic synthesis using nitrilimines. Part 13: synthesis of new
1,2,3,4-Tetrahydro-s-Tetrazine derivatives. Tetrahedron 65:8722–8726
155. Thaher BA, Otto H-H (2002) On the Synthesis of 2-Acetyl-4-aryl-6H-1,3,4-thiadiazin-5-ones
by reaction of nitrilimines with α-mercapto alkanoic acids. Monatshefte für Chemie/ Chem
Mon 133:1011–1016
156. Zahra JA, Abu Thaher BA, El-Abadelah MM, Boese R (2003) An alternative synthesis of
2-(N-Arylhydrazono)-1-benzothiophen-3-ones. Org Biomol Chem 1:822–825
157. Zahra JA, Thaher BA, El-Abadelah MM, Otto H-H (2005) On the synthesis of
some 2-arylhydrazono-3-oxothieno[2,3-b]pyridines by reaction of nitrilimines with 2mercaptonicotinic acid. Monatsh Chem 136:567–570
158. Zahra JA, Abu Thaher BA, El-Abadelah MM, Boese R (2005) 3-mercaptopropionic acid–
nitrile imine adducts. An unprecedented cyclization into 1,3,4-thiadiazol-2(3H)-ones and
-2(3H)-thiones. Org Biomol Chem 3:2599
159. Bruché L, Garanti L, Zecchi G (1981) Intramolecular cyclisations of nitrile imines bearing a
thioether function. J Chem Soc, Perkin Trans 1:2245–2249
160. Bruché L, Garanti L, Zecchi G (1984) New features in the intramolecular capture of nitrile
imines by the sulphide function. J Chem Soc, Perkin Trans 1:2535–2539
161. Meier Hansruedi, Heinzelmann Willy, Heimgartner H (1980) Inter- and intramolecular
trapping reactions of photochemically generated diarylnitrilimines. Chimia (Aarau) 34:506–
508
162. Zhao S, Dai J, Hu M, Liu C, Meng R, Liu X, Wang C, Luo T (2016) Photo-induced coupling
reactions of tetrazoles with carboxylic acids in aqueous solution: application in protein
labelling. Chem Commun 52:4702–4705
163. Herner A, Marjanovic J, Lewandowski TM, Marin V, Patterson M, Miesbauer L, Ready D,
Williams J, Vasudevan A, Lin Q (2016) 2-Aryl-5-carboxytetrazole as a new photoaffinity
label for drug target identification. J Am Chem Soc 138:14609–14615
164. Heiler C, Offenloch JT, Blasco E, Barner-Kowollik C (2017) Photochemically induced folding
of single chain polymer nanoparticles in water. ACS Macro Lett 6:56–61
165. Konrad W, Fengler C, Putwa S, Barner-Kowollik C (2019) Protection-group-free synthesis
of sequence-defined macromolecules via precision λ-orthogonal photochemistry. Angew
Chemie Int Ed 58:7133–7137
